李亦舟Title:博士/教授,博导,硕导 E-mail Address:yizhouli@cqu.edu.cn Tel.:023-65678465 |
2021.07-至今 bat365,副经理
2019.03-至今 bat365•bat365,教授(博士生导师)
2021年获重庆市优秀党务工作者,重庆青年五四奖章
2017.09-2019.02 bat365•bat365,bat365在线登录网站特聘研究员(博士生导师)
2014.09-2017.08 瑞士苏黎世联邦理工大学(ETH),药学博士后,合作导师:Prof. Dario Neri
2009.09-2014.07 北京大学,有机化学专业,理学博士,导师:李笑宇研究员
2005.09-2009.07 北京大学,化学专业,理学学士,导师:施章杰教授
药学化员工物学,化学遗传学,药物分析,中药现代化
以核酸编码化合库(DNA-encoded library)筛选技术为手段的新药先导化合物研究;
以核酸作为工具的化员工物学研究;
对生物大分子的选择性化学修饰;
活性小分子探针设计、合成及靶点识别。
国家自然科学基金委员会优秀青年科学基金项目,2023-01至2025-12,主持,在研
北京分子科学国家研究中心开放课题,2022-01至2023-12,主持,在研
重庆市杰出青年基金项目,2020-09至2023-08,主持,在研
国家自然科学基金委员会青年科学基金项目,2020-01至2022-12,主持,已结题
1.Li Xianfeng#; Zhang Juan#; Liu Changyang; Sun Jie; Li Yangfeng; Zhang Gong*; Li Yizhou*, Aryl Diazonium Intermediates Enable Mild DNA-Compatible C-C Bond Formation for Medicinally Relevant Combinatorial Library Synthesis, Chemical Science, 2022, 13(44): 13100-13109
2.Yang Shilian#; Zhao Guixian#; Gao Yuting; Sun Yang; Fan Xiaohong; Zhang Gong; Li Yangfeng*; Li Yizhou*, In-Solution Direct Oxidative Coupling for the Integration of Sulfur /Selenium into DNA-Encoded Chemical Libraries, Chemical Science, 2022, 13, 2604-2613 (IF= 9.8)
3.Zhao Guixian#; Zhong Shuting#; Zhang Gong; Li Yangfeng; Li Yizhou*, Reversible covalent headpiece enables interconversion between double‐and single‐stranded DNA‐encoded chemical libraries, Angewandte Chemie International Edition, 2022, 61, e202115157 (1 of 7) (IF= 15.3)
4.Huang Yiran; Li Yizhou*; Li Xiaoyu*, Strategies for developing DNA-encoded libraries beyond binding assays, Nature Chemistry, 2022, 14(2): 129-140 (IF= 24.4)
5.Huang Yiran; Meng Ling; Nie Qigui; Zhou Yu; Chen Langdong; Yang Shilian; Fung Yi Man Eva; Li Xiaomeng; Huang Cen; Cao Yan*; Li Yizhou*; Li Xiaoyu*, Selection of DNA-encoded chemical libraries against endogenous membrane proteins on live cells, Nature Chemistry, 2021, 13(1): 77-88 (IF= 24.4)
6.Li Yizhou*; De Luca Roberto; Cazzamalli Samuele; Pretto Francesca; Bajic Davor; Scheuemann Jörg*; Neri Dario*, Versatile protein recognition by the encoded display of multiple chemical elements on a constant macrocyclic scaffold, Nature Chemistry, 2018, 10(4): 441-448 (IF= 24.4)